A Dose Escalation Study of FP-045 in Patients with Fanconi Anemia

Description

This is a multi-center, Phase 1/2 study to determine the Optimal Biologic Dose (OBD) and to evaluate the safety, tolerability, PK, and preliminary activity of FP 045 when administered orally in young adult/adolescent and pediatric patients with Fanconi anemia. The study will enroll a total of 4 young adult/adolescent patients and a minimum of 8 and up to 12 pediatric patients with mild-moderate bone marrow failure who have not undergone hematopoietic cell transplant. This makes the total patient number between 12-16 total. Dose escalation will occur individually for each patient, within each age group. Each patient will receive each of 3 dose levels of FP 045 (intra-patient dose escalation), beginning with Dose Level 1, followed by Dose Levels 2 and 3. Each dose level will be administered for 28 days prior to escalation to the next higher dose level for that patient.

Conditions

Fanconi Anemia

Study Overview

Study Details

Study overview

This is a multi-center, Phase 1/2 study to determine the Optimal Biologic Dose (OBD) and to evaluate the safety, tolerability, PK, and preliminary activity of FP 045 when administered orally in young adult/adolescent and pediatric patients with Fanconi anemia. The study will enroll a total of 4 young adult/adolescent patients and a minimum of 8 and up to 12 pediatric patients with mild-moderate bone marrow failure who have not undergone hematopoietic cell transplant. This makes the total patient number between 12-16 total. Dose escalation will occur individually for each patient, within each age group. Each patient will receive each of 3 dose levels of FP 045 (intra-patient dose escalation), beginning with Dose Level 1, followed by Dose Levels 2 and 3. Each dose level will be administered for 28 days prior to escalation to the next higher dose level for that patient.

A Multinational, Multicenter, Dose Escalation Study to Evaluate the Safety, Tolerability, Pharmacokinetics, and Preliminary Activity of FP 045 in Patients with Fanconi Anemia (FusuciA Study)

A Dose Escalation Study of FP-045 in Patients with Fanconi Anemia

Condition
Fanconi Anemia
Intervention / Treatment

-

Contacts and Locations

Palo Alto

Lucille Packard Children's Hospital, Stanford University, Palo Alto, California, United States, 94305

Minneapolis

Masonic Cancer Center, University of Minnesota, Minneapolis, Minnesota, United States, 55455

New York

David H. Koch Center for Cancer Care at Memorial Sloan Kettering Cancer Center, New York, New York, United States, 10022

Participation Criteria

Researchers look for people who fit a certain description, called eligibility criteria. Some examples of these criteria are a person's general health condition or prior treatments.

For general information about clinical research, read Learn About Studies.

Eligibility Criteria

  • * male or female aged 3-35
  • * documented Fanconi anemia by chromosome breakage analysis
  • * females of child-bearing potential and males required to use highly effective birth control
  • * mild to moderate bone marrow failure with at least one cytopenia of \> grade 1 severity
  • * history of any malignancy except focal squamous cell or basal cell carcinoma of the skin or carcinoma in situ of cervix
  • * has myelodysplastic syndrome or acute leukemia per world health organization (WHO) criteria
  • * has history of any significant medical conditions
  • * has aspartate aminotransferase (AST)/alanine aminotransferase (ALT) \> 5x upper limit of normal (ULN) or calculated creatinine clearance (Clcr) of \< 50 mL/min
  • * has active Hepatitis B or C
  • * has an ongoing systemic infection
  • * requires a strong CYP3A4 inhibitor
  • * has had major surgery within 30 days
  • * Active graft versus host disease requiring systemic treatment
  • * Has a history of bone marrow or stem cell transplant

Ages Eligible for Study

3 Years to 35 Years

Sexes Eligible for Study

ALL

Accepts Healthy Volunteers

No

Collaborators and Investigators

Foresee Pharmaceuticals Co., Ltd.,

Susan Whitaker, STUDY_DIRECTOR, Foresee Pharmaceuticals

Study Record Dates

2025-12